Search results for "VITRO"

showing 10 items of 2786 documents

Synthesis and biological evaluation of novel peptidomimetics as rhodesain inhibitors

2016

Novel rhodesain inhibitors were developed by combining an enantiomerically pure 3-bromoisoxazoline warhead with a 1,4-benzodiazepine scaffold as specific recognition moiety. All compounds were proven to inhibit rhodesain with Ki values in the low-micromolar range. Their activity towards rhodesain was found to be coupled to an in vitro antitrypanosomal activity, with IC50 values ranging from the mid-micromolar to a low-micromolar value for the most active rhodesain inhibitor (R,S,S)-3. All compounds showed a good selectivity against the target enzyme since all of them were proven to be poor inhibitors of human cathepsin L. Novel rhodesain inhibitors were developed by combining an enantiomeri…

rhodesainPharmacologychemistry.chemical_classificationCathepsinPeptidomimetic010405 organic chemistryChemistryPeptidomimeticProton Magnetic Resonance SpectroscopyenPeptidomimetics; rhodesain; trypanosomaGeneral Medicine01 natural sciencesCombinatorial chemistryIn vitro0104 chemical sciencesCysteine Endopeptidases010404 medicinal & biomolecular chemistryEnzymeDrug DiscoveryIc50 valuesMoietyPeptidomimeticsCarbon-13 Magnetic Resonance SpectroscopytrypanosomaBiological evaluationJournal of Enzyme Inhibition and Medicinal Chemistry
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Cryopreservation of Hazelnut (Corylus avellana L.) Axillary Buds from In Vitro Shoots Using the Droplet Vitrification Method

2021

Cryopreservation by droplet vitrification was applied to hazelnut (Corylus avellana L.). axillary buds of the Italian cultivated variety Tonda Gentile Romana, which were collected from in vitro growing shoots, immersed in ice cooled PVS2 or PVS3 for 60 or 90 min, then transferred to a droplet of vitrification solution, placed on a strip of aluminium foil, and plunged into liquid nitrogen (LN). Additionally, the effect on the recovery of the mother plant after cryopreservation was evaluated, following a cold pre-treatment at 4 °C for 3 months. The highest regrowth percentage (56.7%) was obtained after applying PVS3 for 60 min, while the application of PVS2 for the same amount of time reduced…

rootingChemistrylength of dehydrationPlant cultureregrowthPlant ScienceHorticultureLiquid nitrogen<i>in vitro</i> cultureCryopreservationSB1-1110Settore AGR/03 - Arboricoltura Generale E Coltivazioni ArboreeHorticultureAluminium foilAxillary budin vitro cultureShootPVS3PVS2VitrificationHorticulturae
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Cytotoxic Effect of Eudesmanolides Isolated from Flowers of Tanacetum vulgare ssp. siculum

2012

WOS: 000306752700042

sesquiterpeneeudesmanolidePharmaceutical ScienceFlowersSesquiterpeneArticleChinese hamsterCell LineAnalytical ChemistryHuman lungInhibitory Concentration 50Tanacetumchemistry.chemical_compoundsesquiterpenesDrug DiscoveryBotanymedicineAnimalsHumansCytotoxic T cellSettore BIO/15 - Biologia FarmaceuticaPhysical and Theoretical ChemistryTanacetum vulgarecytotoxic activityCell ProliferationCell DeathbiologyTraditional medicine<em>Tanacetum vulgare</em>; sesquiterpenes; eudesmanolides; cytotoxic activityeudesmanolidesOrganic ChemistrySettore CHIM/06 - Chimica Organicabiology.organism_classificationIn vitroTanacetum vulgare; sesquiterpenes; eudesmanolides; cytotoxic activitymedicine.anatomical_structurechemistryPhytochemicalChemistry (miscellaneous)Molecular MedicineColorimetryFormazanMolecules; Volume 17; Issue 7; Pages: 8186-8195
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Propagazione in vitro e produzione di semi sintetici di Metrosoderos excelsa

2009

shoot multiplication ex vitro rooting synthetic seed
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Efectos de un programa de intervención psicoeducativa en la calidad de vida de los/las pacientes durante sus tratamientos de Reproducción Asistida

2021

El término Infertilidad Humana se refiere a la no consecución del embarazo después de 12 meses de mantener relaciones sexuales sin el uso de métodos anticonceptivos. Ha sido reconocido por la Organización Mundial de la Salud (OMS) como un problema de salud pública a nivel global, y aunque existe un alto número de personas con infertilidad, aproximadamente tan sólo la mitad de estas personas buscan tratamientos médicos para lograr concebir. Las personas que se someten a Tratamientos de Reproducción Asistida (TRA) pasan por una serie de etapas en las que sufren distintos tipos de cambios, tanto en su estado físico como emocional. La literatura muestra que durante los tratamientos las mujeres …

sintomatología depresivaintervención psicológicapsicología ansiosafecundación in vitropsicología clínica:PSICOLOGÍA [UNESCO]UNESCO::PSICOLOGÍAevaluación psicológicainfertilidadreproducción asistidaajuste psicológicoestrés emocionalabordaje psicológico en infertilidadapoyo socialintervención psicoeducativacalidad de vidapsicología de la saludestimulación hormonalcuidado psicosocial
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Morphological and Anatomical Observations of Abnormal Somatic Embryos from Anther Cultures of Citrus reticulata Blanco.

2010

somatic embryogenesis mandarinanatomy in vitro cultureCitrus in vitro culture
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Optical quality of hyperopic and myopic phakic intraocular lenses

2013

Aims: To assess and compare the optical quality of the myopic and hyperopic implantable collamer lens (ICL) from its wavefront aberrations for different powers and pupil diameters. Settings and Design: Prospective study. Material and Methods: The wavefront aberrations of two myopic (−3 and −6 diopters (D)) and two hyperopic V4b ICLs (+3 and +6D) were measured in vitro . To assess and compare the optical quality of different powers of ICLs, we analyzed the root mean square (RMS) of total higher order aberrations (HOAs), trefoil, coma, tetrafoil, secondary astigmatism, and spherical aberration at 3- and 4.5-mm pupil. In addition, the point spread functions (PSFs) of each ICL evaluated were ca…

steep corneal curvatureintravitreallacrimal fossaRefractive errorvisual acuitygenetic structurespterygium surgerystandard automated perimetryComa (optics)BlindnessPhakic intraocular lenslaw.inventionsubconjunctival bevacizumab injectionCorneaLens Implantation Intraocularlcsh:Ophthalmologylawmodified deep anterior lamellar keratoplastyMitomycin CMaterials TestingAutogenous tissue graftingProspective StudiesDioptreoptical qualityshort wave automated perimetryexcimer lasernon-proliferative diabetic retinopathyMean deviationin vitroheavy silicone oilBevacizumabLens (optics)Aberrations of the eyeSpherical aberrationHyperopiaAntimicrobial effectOriginal ArticleTriamcinolone acetonidehuman trabecular meshwork cellsPhakic Intraocular Lensesmedicine.medical_specialtyImaging in glaucomadisability evaluationconventional silicone oiltriamcinoloneProsthesis DesignKeratoconusphotorefractive keratectomyOphthalmologygrowth factorsmedicineHumansmyopiamyopic implantable collamer lensshort fluctuationsWavefrontmacular edemaoptical coherence tomographyendophthalmitis agentsbusiness.industrybranch retinal vein occlusionretinal nerve fiber layerpterygium recurrencemedicine.diseaseeye diseasesOphthalmologypediatricwavefront aberrationsquality of lifelcsh:RE1-994bypass surgeryHyperopic implantable collamer lenslacrimal drainage systemsense organsbusinessIndian Journal of Ophthalmology
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Drought Stress Study on Nicotiana tabacum L., “Baladi”, an In Vitro Experimental Model

2021

Crops drought tolerance is a trait of outmost importance for agriculture especially today when climate change is affecting more the production for food and feed. The scope of this article is to evaluate in vitro drought stress response of Nicotiana tabacum L., “Baladi”. The experiment was set up for four successive stages starting with in vitro seedling development, hypocotyl cultivation, three generations of micropropagation, pre-acclimatization and acclimatization. The effect of abscisic acid (ABA) and/or polyethylene-glycol 6000 (PEG) on tobacco hypocotyl caulogenesis and micropropagation were investigated. Superoxide-dismutases (SODs) and peroxidases (POXs) are more active and different…

superoxide-dismuthaseAgriculture (General)Nicotiana tabacumDrought toleranceperoxidasedroughtPlant SciencetobaccoAcclimatizationS1-972Hypocotylchemistry.chemical_compoundhypocotylsAbscisic acidbiologyfungifood and beveragesin vitrobiology.organism_classificationacclimatizationshootingHorticulturechemistryMicropropagationSeedlingShootAgronomy and Crop ScienceFood ScienceAgriculture
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Water-Soluble Cuprizone Derivative: Synthesis, Characterization, and in Vitro Studies

2019

The cuprizone mouse model is one of the most accepted model systems for the investigation of oligodendrocyte degeneration, a process critically involved in the pathogenesis of diseases such as multiple sclerosis or schizophrenia. In order to substitute the in vivo experiments by in vitro approaches, the amine derivative BiMPi is introduced as a water-soluble alternative to cuprizone. Regarding superoxide dismutase activity, toxicity for oligodendrocytes, and disturbance of mitochondrial membrane potential, BiMPi shows similar in vitro effects as is observed in vivo for cuprizone. peerReviewed

synthesispatogeneesiGeneral Chemical EngineeringDegeneration (medical)010402 general chemistry01 natural sciencesneurokemialcsh:ChemistryPathogenesis03 medical and health scienceschemistry.chemical_compound0302 clinical medicinemedicinecharacterizationsynteesita116water-soluble cuprizone derivativekemiallinen synteesiin Vitro studiesamiinitChemistryta1182General ChemistryOligodendrocyteIn vitro3. Good health0104 chemical sciencesmedicine.anatomical_structureWater solublelcsh:QD1-999Biochemistryin vitro -menetelmä030217 neurology & neurosurgeryDerivative (chemistry)
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No Dracocephalum ruyschiana L. iegūtu bioloģiski aktīvo vielu ādu balinošo īpašību novērtējums in vitro

2016

Darba mērķis bija novērtēt no Ruiša pūķgalves savvaļas augiem un in vitro dzinumu kultūrām iegūtu bioloģiski aktīvos savienojumus saturošu ekstraktu ādu balinošās īpašības, izmantojot in vitro testēšanas metodes. Ruiša pūķgalves in vitro ekstrakta drošība tā pielietojumam kosmētikas preparātos tika noteikta, pārbaudot tā ietekmi uz dažādu ādas tipu šūnu proliferāciju un morfoloģiju. Ādu balinošā potenciāla novērtēšanai tika izmantots sēņu tirozināzes inhibīcijas tests un cilvēka ādas melanomas šūnu in vitro modelis. No Ruiša pūķgalves in vitro dzinumu kultūras tika iegūts savvaļas augam līdzvērtīgs un lietošanai drošs ekstrakts, kas inhibēja sēņu un šūnu tirozināzes aktivitāti, bet būtisiki…

tirozināzein vitro testēšanaādu balinošā kosmētikaRuiša pūķgalveaugu in vitro kultūrasBioloģija
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