Search results for "ivermectin"

showing 10 items of 16 documents

Microscopic interactions between ivermectin and key human and viral proteins involved in SARS-CoV-2 infection

2021

The identification of chemical compounds able to bind specific sites of the human/viral proteins involved in the SARS-CoV-2 infection cycle is a prerequisite to design effective antiviral drugs. Here we conduct a molecular dynamics study with the aim to assess the interactions of ivermectin, an antiparasitic drug with broad-spectrum antiviral activity, with the human Angiotensin-Converting Enzyme 2 (ACE2), the viral 3CLpro and PLpro proteases, and the viral SARS Unique Domain (SUD). The drug/target interactions have been characterized in silico by describing the nature of the non-covalent interactions found and by measuring the extent of their time duration along the MD simulation. Results …

DrugProteasesIn silicomedia_common.quotation_subjectProtein domainCoronavirus Papain-Like ProteasesGeneral Physics and AstronomyPlasma protein bindingBiologyAntiviral AgentsivermectinProtein DomainsMolecular dynamics simulationHumansPhysical and Theoretical ChemistryBinding siteCoronavirus 3C Proteasesmedia_commonchemistry.chemical_classificationSARS Unique DomainBinding SitesSARS-CoV-2SARS-CoV-2 infectionRNAHydrogen BondingVirologyG-QuadruplexesMolecular Docking SimulationEnzymechemistrySettore CHIM/03 - Chimica Generale E InorganicaRNAAngiotensin-Converting Enzyme 2Hydrophobic and Hydrophilic InteractionsProtein BindingPhysical Chemistry Chemical Physics
researchProduct

Donor-derived Strongyloides stercoralis hyperinfection syndrome after simultaneous kidney/pancreas transplantation

2016

Most cases of strongyloidiasis associated with solid organ transplantation have been due to the reactivation of a latent infection in the recipient as a result of the immunosuppressive therapy; however, donor-derived infections are becoming increasingly frequent. The case of a patient who nearly died of a Strongyloides stercoralis hyperinfection after receiving simultaneous kidney/pancreas transplants is described herein. No specific parasitological tests were performed pre-transplantation, despite the fact that both the recipient and the donor originated from endemic areas. Serological analysis of the donor's serum performed retrospectively revealed the origin of the infection, which if it…

Microbiology (medical)AdultMalemedicine.medical_specialtymedicine.medical_treatment030231 tropical medicineHyperinfection030230 surgeryPancreas transplantationTransplantKidneyGastroenterologylcsh:Infectious and parasitic diseasesStrongyloides stercoralisSerology03 medical and health sciences0302 clinical medicineDonor-derivedAparell urinariInternal medicineStrongyloidesmedicineAnimalsHumanslcsh:RC109-216PancreasKidney transplantationImmunosuppression TherapyIvermectinbiologybusiness.industryImmunosuppressionGeneral Medicinebiology.organism_classificationmedicine.diseaseKidney TransplantationTissue DonorsSurgeryTransplantationInfectious DiseasesStrongyloidiasisStrongyloidesInfeccióStrongyloidiasisPancreas TransplantationbusinessStrongyloides stercoralis
researchProduct

Case report: Control of intestinal nematodes in captive Chlorocebus sabaeus

2021

Funding was provided by the Ross University School of Veterinary Medicine via the One Health Center for Zoonoses and Tropical Veterinary Medicine.

MaleVeterinary medicineTrichurisTrichostrongyluscapillariaNematodesVeterinary medicine0403 veterinary scienceFeces0302 clinical medicineIvermectinChlorocebus aethiopsSF600-1100StrongyloidesCaptiveTrichostrongylusAnthelminticseducation.field_of_studybiology04 agricultural and veterinary sciencesGeneral MedicineTrichurishookwormmedicine.drugHookworm040301 veterinary sciences030231 tropical medicinePopulationCapillariaafrican green monkeysalbendazoleAfrican green monkeyscaptiveAlbendazoleAlbendazoleivermectinResearch Communication03 medical and health sciencesstrongyloidesparasitic diseasesmedicineAnimalsTrichuriasiseducationParasite Egg CountIvermectinGeneral VeterinarytrichurisParasitologia veterinàriabiology.organism_classificationStrongyloidesCapillariaTrichuris trichiuratrichostrongylus
researchProduct

Effect of ivermectin on the liver of gilthead sea bream Sparus aurata: a proteomic approach.

2010

23 p., 2 tablas, 4 figuras y bibliografía

ProteomicsFish ProteinsEnvironmental EngineeringNew biomarkersSparidaeProteomeHealth Toxicology and MutagenesisDifference gel electrophoresisBiologyIvermectinAquaculturemedicineEnvironmental ChemistryAnimalsGilthead seabreamIvermectinAntiparasitic AgentsEcologybusiness.industryPublic Health Environmental and Occupational HealthHepatotoxinLipid metabolismAquatic animalGeneral MedicineGeneral ChemistryMetabolismbiology.organism_classificationPollutionSea BreamMass spectrometry (MS)BiochemistryLiver2D-DIGEbusinessBiomarkersWater Pollutants Chemicalmedicine.drugChemosphere
researchProduct

In Vitro Testing of Alternative Synthetic and Natural Antiparasitic Compounds against the Monogenean Sparicotyle chrysophrii

2021

© 2021 by the authors.

Microbiology (medical)AnthelminthicsAntiparasiticmedicine.drug_class<i>Sparicotyle chrysophrii</i>AquacultureBiologyMicrobiology03 medical and health sciencesIvermectinAquacultureSettore AGR/20 - Zoocolturemedicinegilthead sea breamImmunology and AllergyParasite hostingPotency14. Life underwateranthelminthicsMolecular Biology030304 developmental biology0303 health sciencesGeneral Immunology and MicrobiologyVibrio harveyibusiness.industryR04 agricultural and veterinary sciencesanthelminthics ; aquaculture ; gilthead sea bream ; monogenea ; Sparicotyle chrysophriimonogeneabiology.organism_classification3. Good healthPraziquantelInfectious DiseasesaquacultureGilthead sea breamSparicotyle chrysophriiToxicity040102 fisheries0401 agriculture forestry and fisheriesMedicinebusinessMonogeneamedicine.drugPathogens
researchProduct

Experimental infection of the deer ked (Lipoptena cervi) has no negative effects on the physiology of the captive reindeer (Rangifer tarandus tarandu…

2011

The deer ked (Lipoptena cervi) is a haematophagous parasitic fly of cervids that spread to Finland in the early 1960's. Presently its northern distribution limit lies at approximately 65°N and it is gradually spreading northwards. In Finland the principal host species has been the moose (Alces alces), but the deer ked is about to establish contact with another potential host, the semi-domesticated reindeer (Rangifer tarandus tarandus) causing possible threats to reindeer health and management. The aim of this study was to investigate if the deer ked would have an influence on the welfare of the reindeer. Eighteen adult reindeer were divided into three experimental groups: the control group …

Male0106 biological sciencesInsecticidesVeterinary medicineParasitismEctoparasitic Infestations010603 evolutionary biology01 natural sciences03 medical and health sciencesIvermectinbiology.animalmedicineAnimals030304 developmental biology0303 health sciencesIvermectinGeneral VeterinarybiologyHippoboscidaeHost (biology)DipteraGeneral Medicinebiology.organism_classificationPhysiological AdaptationsRangifer tarandus tarandus13. Climate actionLipoptena cerviFemaleParasitologyReindeermedicine.drugVeterinary Parasitology
researchProduct

The prevalence of onchocerciasis in Africa and Yemen, 2000-2018: a geospatial analysis.

2022

Abstract Background Onchocerciasis is a disease caused by infection with Onchocerca volvulus, which is transmitted to humans via the bite of several species of black fly, and is responsible for permanent blindness or vision loss, as well as severe skin disease. Predominantly endemic in parts of Africa and Yemen, preventive chemotherapy with mass drug administration of ivermectin is the primary intervention recommended for the elimination of its transmission. Methods A dataset of 18,116 geo-referenced prevalence survey datapoints was used to model annual 2000–2018 infection prevalence in Africa and Yemen. Using Bayesian model-based geostatistics, we generated spatially continuous estimates o…

Onchocerciasis; Geospatial model; Neglected tropical diseases;IvermectinYemenSettore MED/06 - Oncologia MedicaSettore MED/42 - Igiene Generale e ApplicataNigeriaBayes TheoremGeneral MedicineOnchocerciasisGhanaSettore MED/01 - Statistica MedicaGeneral & Internal MedicinePrevalenceHumansGeospatial model11 Medical and Health SciencesNeglected tropical diseasesBMC medicine
researchProduct

Comparison between whole-body MRI with diffusion-weighted imaging and PET/CT in staging newly diagnosed FDG-avid lymphomas.

2015

Abstract Objectives To compare whole body-MRI (WB-MRI) with diffusion-weighted imaging and FDG-PET/CT in staging newly diagnosed FDG-avid lymphomas. Methods 68 patients (37 males, 31 females; median age 42 years; range 15–86 years) with histologically confirmed lymphoma (37 Classical Hodgkin, 16 Diffuse large B-cell, 10 Follicular, 5 Mantle cell) underwent both MRI and FDG-PET/CT before treatment. Ann Arbor stages obtained with WB-MRI and FDG-PET/CT were compared using Cohen’s k statistics. Moreover WB-MRI and FDG-PET/CT stages were compared with the pathological stages obtained after the diagnostic iter using also bone marrow and available biopsies if clinically indicated. Results The agre…

MaleStagingLymphomaMultimodal Imaging030218 nuclear medicine & medical imaging0302 clinical medicineWhole Body ImagingProspective StudiesStage (cooking)Computed tomographyAged 80 and overmedicine.diagnostic_testGeneral MedicineMiddle AgedPositron emission tomography030220 oncology & carcinogenesisRadiopharmaceuticalFemaleDiffusion-weighted imagingRadiologyHumanmedicine.drugAdultmedicine.medical_specialtyAdolescentWhole body imagingReproducibility of ResultYoung Adult03 medical and health sciencesMagnetic resonance imagingFluorodeoxyglucose F18medicineHumansRadiology Nuclear Medicine and imagingAgedNeoplasm StagingFluorodeoxyglucosePET-CTIvermectinbusiness.industryReproducibility of ResultsMagnetic resonance imagingmedicine.diseaseLymphomaProspective StudieDiffusion Magnetic Resonance ImagingPositron-Emission TomographyMantle cell lymphomaRadiopharmaceuticalsSettore MED/36 - Diagnostica Per Immagini E RadioterapiaTomography X-Ray ComputedNuclear medicinebusinessEuropean Journal of Radiology
researchProduct

Determination of abamectin in citrus fruits by liquid chromatography-electrospray ionization mass spectrometry.

2000

Liquid chromatography coupled to electrospray mass spectrometry (LC-ES-MS) with positive ion detection was used to determine abamectin in oranges. MS conditions were optimized to achieve maximum sensitivity. The main ion for abamectin was [M+Na]+ at a fragmentor voltage of 180 V. Abundant structural information can be obtained at different fragmentor voltages. The detection limit for the standard solution was 12 pg injected, and good linearity and reproducibility were observed. Abamectin residues were extracted using matrix solid-phase dispersion. Orange samples were homogenized with C18 bonded silica placed onto a glass column and eluted with dichloromethane. Recoveries of the abamectin fr…

Detection limitQuality ControlElectrosprayCitrusInsecticidesChromatographyIvermectinElutionElectrospray ionizationOrganic ChemistryReproducibility of ResultsGeneral MedicineMass spectrometryBiochemistryHigh-performance liquid chromatographySensitivity and SpecificityMass SpectrometryAnalytical Chemistrychemistry.chemical_compoundchemistryAbamectinSolid phase extractionChromatography High Pressure LiquidJournal of chromatography. A
researchProduct

Predicting the environmental suitability for onchocerciasis in Africa as an aid to elimination planning

2021

Recent evidence suggests that, in some foci, elimination of onchocerciasis from Africa may be feasible with mass drug administration (MDA) of ivermectin. To achieve continental elimination of transmission, mapping surveys will need to be conducted across all implementation units (IUs) for which endemicity status is currently unknown. Using boosted regression tree models with optimised hyperparameter selection, we estimated environmental suitability for onchocerciasis at the 5 × 5-km resolution across Africa. In order to classify IUs that include locations that are environmentally suitable, we used receiver operating characteristic (ROC) analysis to identify an optimal threshold for suitabil…

OncocercosisDecision AnalysisRC955-962Onchocerciasislaw.inventionGeographical LocationsMedical Conditions0302 clinical medicinelawArctic medicine. Tropical medicineMedicine and Health Sciences030212 general & internal medicineOnchocerca11 Medical and Health SciencesData ManagementbiologyPharmaceuticswc_695Enfermedades ParasitariasOnchocerciasi3. Good healthInfectious DiseasesGeographyTransmission (mechanics)Helminth InfectionsEngineering and TechnologyMass Drug AdministrationOnchocercaPublic aspects of medicineRA1-1270Management EngineeringCartographyHumanResearch ArticleNeglected Tropical DiseasesComputer and Information SciencesDrug Administration030231 tropical medicineDecision treewa_395Dermatologywc_765Environmentwc_885Research and Analysis MethodsSkin Diseases03 medical and health sciencesDrug TherapySDG 3 - Good Health and Well-beingDiagnostic MedicineTropical MedicineParasitic DiseasesmedicineHumansDisease EradicationSpatial analysisIvermectinData collectionReceiver operating characteristicData VisualizationDecision TreesPublic Health Environmental and Occupational Health06 Biological SciencesOnchocerciasis ; Elimination planning ; Africa ; Implementation units ; Public healthTropical Diseasesmedicine.diseasebiology.organism_classificationHealth CareROC CurvePeople and PlacesAfricaHealth StatisticsMorbidityOnchocerciasisScale (map)ForecastingPLOS Neglected Tropical Diseases
researchProduct