Search results for "magnetic resonance spectroscopy"

showing 10 items of 1362 documents

Installation of Amine Moieties into a Polycyclic Anodic Product Derived from 2,4-Dimethylphenol

2011

When 2,4-dimethylphenol is anodically treated, a dehydrotetramer with four contiguous stereocentres is readily obtained on a multi-gram scale. The substitution of a 2,4-dimethyl-phenoxy fragment by several amines was demonstrated, and the best results were obtained with primary amines. Optically pure α-chiral aliphatic amines yield diastereomeric mixtures that can be separated in most cases. The basic amine causes a partial hemiketal-opening of the bisbenzofuran moiety leading to an equilibrium within an α,β-unsaturated cyclohexenone. This dynamic behaviour occurs on the time scale of NMR spectroscopy and is also found by X-ray analysis providing a consistent picture.

ChemistryOrganic ChemistryDiastereomerGeneral ChemistryNuclear magnetic resonance spectroscopyCatalysisChiral resolutionchemistry.chemical_compoundCyclohexenoneYield (chemistry)MoietyOrganic chemistryAmine gas treatingAminationChemistry - A European Journal
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5-Alkenyl-1,2,3-thiadiazole

1986

Es wird die Herstellung der Titelverbindungen 5 durch Bromierung-Dehydrobromierung entsprechender 5-Alkyl-1,2,3-thiadiazole 3, ihre spektroskopische Charakterisierung und ihre Umsetzung mit 4-Phenyl-4H-1,2,4-triazol-3,5-dion (6) zu 7, 8 beschrieben. 5-Alkenyl-1,2,3-thiadiazoles A method of preparation for the title compounds 5, by bromination-dehydrobromination of the corresponding 5-alkyl-1,2,3-thiadiazoles 3, their spectroscopical characterization, and the reaction of 5 with 4-phenyl-4H-1,2,4-triazole-3,5-dione (6) with formation of 7, 8 is described.

ChemistryOrganic ChemistryHalogenationNuclear magnetic resonance spectroscopyPhysical and Theoretical ChemistryMedicinal chemistryCycloadditionLiebigs Annalen der Chemie
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Determination of the Relative Stereochemistry of Flexible Organic Compounds by Ab Initio Methods: Conformational Analysis and Boltzmann-Averaged GIAO…

2002

Ab initio calculations at the Hartree-Fock level with full-geometry optimization using the 6-31G(d) basis set, and GIAO (gauge including atomic orbitals) 1 3 C NMR chemical shifts, are presented here as a support in the study of the stereochemistry of low-polar organic compounds having an openchain structure. Four linear stereoisomers, fragments of a natural product previously characterized by experimental 1 3 C NMR spectra, which possesses three stereogenic centers, 11 carbon atoms, and 38 atoms in total, were considered. Conformational searches, by empirical force-field molecular dynamics, pointed out the existence of 8-13 relevant conformers per stereoisomer. Thermochemical calculations …

ChemistryStereochemistryChemical shiftOrganic ChemistryAb initioGeneral ChemistryNuclear magnetic resonance spectroscopyCarbon-13 NMRCatalysisAb initio quantum chemistry methodsComputational chemistryAtomConformational isomerismBasis setChemistry - A European Journal
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Tautomerism and the Protonation/Deprotonation of Isocytosine in Liquid- and Solid-States Studied by NMR Spectroscopy and Theoretical Calculations

2011

Isocytosine crystallizes as a 1:1 ratio of two tautomers in a manner similar to that of the guanine and cytosine pairs in DNA. The solid-state NMR chemical shifts of crystalline neutral isocytosine, the sodium salt of isocytosine, and those of isocytosine hydrochloride were measured and related to the NMR parameters in aqueous and organic solutions. The experimental chemical shifts were compared with those calculated by three different methods: (1) calculations on isolated molecules, (2) calculations on isocytosine clusters of various sizes, and (3) infinite crystal calculations, that is, the gauge-including projector-augmented wave (GIPAW) method. The data obtained with the GIPAW method we…

ChemistryStereochemistryChemical shiftOrganic ChemistryProtonationNuclear magnetic resonance spectroscopyCrystal structureTautomerchemistry.chemical_compoundDeprotonationMoleculePhysical chemistryIsocytosinePhysical and Theoretical Chemistryta116European Journal of Organic Chemistry
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1H,13C and17O NMR study of aromatic ring-substituted monochloro- and monobromo-(E)-3-phenylpropenals

1991

Trans-Cinnamaldehydes (CAs) or o-, m- and p-X-(E)-3-phenylpropenals; (X = Cl or Br) were synthesized and their 1H, 13C and 17O NMR spectra were measured, assigned and analysed. The long-range benzylic couplings are discussed in terms of the conformational characteristics of the related styrene systems. The 1H, 13C and 17O NMR substituent chemical shifts of the CA derivatives were compared with those of styrene and explained by the π-electron delocalization in the conjugated CCCO bond system of CA.

ChemistryStereochemistryChemical shiftSubstituentGeneral ChemistryNuclear magnetic resonance spectroscopyConjugated systemRing (chemistry)Medicinal chemistryStyrenechemistry.chemical_compoundDelocalized electronGeneral Materials ScienceSolvent effectsMagnetic Resonance in Chemistry
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Antivirale Wirkstoffe, 27. Mitt. Die Aminomethinylierung von 5-Oxo-2-pyrazolin-3-carbonsäurederivaten

1986

Aus der mit s-Triazin (1) durchgefuhrten Aminomethinylierung der 5-Oxo-2-pyrazolin-3-carbonsaurederivate 2a,b gehen die 4-Aminomethylen-5-oxo-2-pyrazolin-3-carbonsaurederivat 4a,b und die C-Rubazonsauren 5a,b hervor. Bei 4a deuten die spektroskopischen Daten auf das Vorliegen der Z-Form (Abb. 1), fur 5a auf das der Z-s-cis-(OH)-Form (Abb. 2) hin. Die Strukturtypen 4 und 5 weisen Vertreter mit antiviraler, entzundungshemmender, temperatursenkender und antimykotischer Wirkung auf. Antiviral Agents, XXVII: Aminomethynylation of 5-Oxo-2-pyrazoline-3-carboxylic Acid Derivatives Aminomethynylation of the 5-oxo-2-pyrazoline-3-carboxylic acid derivatives 2a,b by means of s-triazine (1) yields the 4…

ChemistryStereochemistryDrug DiscoveryMass spectrumPharmaceutical ScienceBiological activityNuclear magnetic resonance spectroscopyArchiv der Pharmazie
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Syntheses, Structures and Reactivity of New Intramolecularly Coordinated Tin Alkoxides Based on an Enantiopure Ephedrine Derivative

2011

The syntheses of the tin compounds [LSn]2 (2), spiro-L2Sn (3), [LSnW(CO)5]2 (4), [LSnBr2]2 (5), spiro-L2Sn·SnBr4 (6) and LSn[OC(O)Ph]2 (8), where L = MeN(CH2CMe2O)[(S)-CH(Me)-(R)-CH(Ph)O], and (Ph4P)2SnBr6 (7) are reported. The compounds were characterized by elemental analysis, multinuclear NMR spectroscopy including 119Sn cross polarisation–magic angle spinning NMR (CP–MAS) (2, 3–6), electrospray ionization mass spectrometry (2–4) and single crystal X-ray diffraction analysis (2, 2·C7H8, 3a, 3b, 4·C7H8, 5, 6·C7H8, 7).

ChemistryStereochemistryElectrospray ionizationchemistry.chemical_elementNuclear magnetic resonance spectroscopyMedicinal chemistryInorganic Chemistrychemistry.chemical_compoundEnantiopure drugElemental analysisReactivity (chemistry)TinSingle crystalDerivative (chemistry)European Journal of Inorganic Chemistry
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1H,13C and17O NMR study of substituted nitropyridines

1991

1H, 13C and 17O NMR spectra for 22 substituted nitropyridines were measured and their 1H NMR spectra were analysed. The most significant variations in the NMR parameters are found for isomeric hydroxy derivatives, owing to the possibility of keto–enol tautomerism. The prevalence of the keto form is observed in 2- and 4-hydroxy derivatives, while the 3-hydroxy derivative exists in its enol form. Among the three nuclei studied, 17O seems to be the best nucleus for probing the keto–enol tautomerism. No correlation is observed between the torsion angle of the nitro group and its 17O NMR chemical shift. Molecular mechanics calculations were performed to clarify the torsional energetics of the ni…

ChemistryStereochemistryGeneral ChemistryKeto–enol tautomerismNuclear magnetic resonance spectroscopyDihedral angleTautomerEnolchemistry.chemical_compoundMolecular dynamicsComputational chemistryNitroProton NMRGeneral Materials ScienceMagnetic Resonance in Chemistry
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Protonation of 3-aminopyrroles

1987

Abstract The protonation of 3-aminopyrroles has been investigated using H and 13C n.m.r. spectroscopy. The spectral data are compatible with predominant protonation of the amino group with no evidence for protonation of the pyrrole ring.

ChemistryStereochemistryNuclear TheoryOrganic ChemistryProtonationNuclear magnetic resonance spectroscopyRing (chemistry)BiochemistryMedicinal chemistrychemistry.chemical_compoundDrug DiscoveryPhysics::Accelerator PhysicsChemical solutionNuclear ExperimentSpectroscopySpectral dataPyrroleTetrahedron
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An experimental and theoretical study of the isomerization of mononuclear bis(arylselenolato)bis(triphenylphosphine)platinum complexes [Pt(SeR)2(PPh3…

2003

Abstract Mononuclear bis(thienylselenolato)bis(triphenylphosphine)platinum [Pt(SeTh)2(PPh3)2] (Th=2-thienyl, C4H3S) has been prepared by the treatment of cis-[PtCl2(PPh3)2] with NaSeTh. The 31P-NMR spectroscopic information indicates that cis-[Pt(SeTh)2(PPh3)2] is initially formed in the reaction. Upon prolonged standing in solution it isomerizes to trans-[Pt(SeTh)2(PPh3)2]. The reaction of cis-[PtCl2(PPh3)2] with LiSeFu (Fu=2-furyl, C4H3O) affords immediately a mixture of cis- and trans-isomers of [Pt(SeFu)2(PPh3)2] with the relative amount of the trans-isomer increasing with time. The recrystallization of the two reaction mixtures yielded cis,anti- and trans,syn-isomers of [Pt(SeTh)2(PPh3…

ChemistryStereochemistryOrganic ChemistryAb initiochemistry.chemical_elementNuclear magnetic resonance spectroscopyBiochemistryMedicinal chemistryInorganic Chemistrychemistry.chemical_compoundX-ray crystallographyMaterials ChemistryMolecular orbitalPhysical and Theoretical ChemistryTriphenylphosphinePlatinumIsomerizationJournal of Organometallic Chemistry
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