Search results for "stigmas"

showing 10 items of 41 documents

Polyamine conjugates of stigmasterol.

2012

Abstract Three new polyamine conjugates with stigmasterol [(3β,22 E )-stigmasta-5,22-dien-3-ol] were synthesized and subjected to basic antimicrobial and cytotoxic tests. The conjugate derived from spermine, (3β,22 E )-stigmasta-5,22-dien-3-yl 4(12-amino-4,9-diaza-dodecylamino)-4-oxobutanoate ( 5c ), displayed considerable antimicrobial activity on Staphylococcus aureus at low concentration (50 μg mL −1 ). The cytotoxic activity was tested on cells of human T-lymfoblastic leukemia (IC 50  = 35.8 ± 10.3 μM ( 5c ) and IC 50  = 35.9 ± 5.7 μM ( 5b )) and normal human fibroblasts (IC 50  = 38.0 ± 2.8 μM ( 5c ) and IC 50  = 45.5 ± 1.9 μM ( 5b )). Conjugate 5a displayed no activity in both tests.

Models MolecularStaphylococcus aureusChemical PhenomenaStereochemistryClinical BiochemistryCarboxylic AcidsMolecular ConformationStigmasterolSpermineAntineoplastic Agentsmedicine.disease_causeBiochemistrychemistry.chemical_compoundEndocrinologyAmideCell Line TumormedicinePolyaminesCytotoxic T cellHumansta116Molecular BiologyPharmacologyStigmasterolDose-Response Relationship DrugOrganic ChemistryAntimicrobialAnti-Bacterial AgentschemistryStaphylococcus aureusDrug DesignPolyamineConjugateSteroids
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Two new sesquiterpene derivatives from the Tunisian endemic Ferula tunetana Pom.

2010

A new sesquiterpene ester, tunetanin A (1), a new sesquiterpene coumarin, tunetacoumarin A (2), together with eight known compounds, i.e., coladin (3), coladonin (4), isosmarcandin (5), 13-hydroxyfeselol (6), umbelliprenin (7) propiophenone (8), beta-sitosterol (9), and stigmasterol (10), were isolated from the roots of Ferula tunetana. Their structures were elucidated on the basis of extensive spectroscopic methods, including 1D- and 2D-NMR experiments and MS analysis, as well as by comparison with published data. The cytotoxicity of compounds 1-7 towards two human colon cancer cell lines, HT-29 and HCT 116, was evaluated. Compounds 3, 4, and 6 showed weak cytotoxic activities.

Magnetic Resonance SpectroscopyStereochemistryBioengineeringSesquiterpeneBiochemistryPlant Rootschemistry.chemical_compoundStructure-Activity RelationshipPropiophenoneSpecies SpecificityCoumarinsCell Line TumorHumansCytotoxicityMolecular BiologyCell ProliferationStigmasterolMs analysisGeneral ChemistryGeneral MedicineCoumarinAntineoplastic Agents PhytogenicUmbellipreninFerulachemistryFerula tunetanaMolecular MedicineDrug Screening Assays AntitumorSesquiterpenesChemistrybiodiversity
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Sterol Composition in Infant Formulas and Estimated Intake.

2015

Sterol contents in infant formulas (IFs) from the European market were determined, and their intakes by infants between 0 and 6 months were evaluated. Total animal sterols (mg/100 mL) ranged from 1.71 to 5.46, cholesterol being the main animal sterol (1.46-5.1). In general, cholesterol and desmosterol were lower than the human milk (HM) values indicated by other authors. Total plant sterol (mg/100 mL) ranged from 3.1 to 5.0. β-Sitosterol, the most abundant phytosterol, ranged from 1.82 to 3.01, followed by campesterol (0.72-1.15), stigmasterol (0.27-0.53), and brassicasterol (0.14-0.28). Cholesterol intake (mg/day) ranged from 9 to 51 and plant sterol intake (mg/day) from 19 to 50. The ster…

StigmasterolMolecular StructureCholesterolCampesterolPhytosterolInfantGeneral ChemistryBrassicasterolBiologySterolInfant Formulachemistry.chemical_compoundSterolschemistryInfant formulaDesmosterolAnimalsHumanslipids (amino acids peptides and proteins)CattleFood scienceGeneral Agricultural and Biological SciencesJournal of agricultural and food chemistry
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Identification of bound alcohols in soil humic acids by gas chromatography-mass spectrometry

2000

International audience; Humic acids are complex, partly macromolecular, yellow-brownish substances occurring in soils, waters and sediments. In order to shed some light on their molecular structure, crop humic acids were cleaved by alkaline hydrolysis (KOH). The products were fractionated by thin layer chromatography to give mono-alcohols which were analysed as acetate derivatives by gas chromatography coupled to mass spectrometry. Linear alcohols, sterols, stanols and plant-derived triterpenoid alcohols were identified by co-injection of pure standards and by comparison with literature data. These findings imply that alcohols could have been incorporated into the humic matrix by esterifica…

[SDE] Environmental SciencescampesterolKOH hydrolysisstanols[SDV]Life Sciences [q-bio]TLCFatty alcoholBrassicasterolAlkaline hydrolysis (body disposal)chemical degradation[SDV.SA.SDS]Life Sciences [q-bio]/Agricultural sciences/Soil study010402 general chemistryMass spectrometry01 natural sciencescomplex mixtureskerogenchemistry.chemical_compoundsterolstigmasterolOrganic chemistrySpectroscopyChromatographyhuminChemistryhumic substancesamyrin010401 analytical chemistrybrassicasterolcholesterolGeneral MedicineAtomic and Molecular Physics and OpticsThin-layer chromatography0104 chemical sciences[SDV] Life Sciences [q-bio]CHIMIE ANALYTIQUEsitosteroln-alkanols[SDE]Environmental SciencesHumintriterpenoidGas chromatographyGas chromatography–mass spectrometryGC-MSfatty alcohol
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Unprecedented new nonadecylpara-hydroperoxycinnamate isolated fromErythrina excelsaand its cytotoxic activity

2014

A new unprecedented cinnamate derivative (1) was obtained from Erythrina excelsa (Leguminosae) and identified as nonadecyl para-hydroperoxycinnamate. This compound was isolated together with three known compounds, namely lupeol (2), mixture of sitosterol and stigmasterol (3), and isoneorautenol (4). Their structures were established on the basis of NMR and mass spectroscopic data in conjunction with those reported in the literature. Compound 1 was evaluated for its capability of inhibiting cancer cell lines and growth of a panel of microbial strains. It turned out that 1 is moderately to significantly cytotoxic against six cancer cell lines and shows weak to no antimicrobial activity.

Magnetic Resonance SpectroscopyStereochemistryPlant ScienceBiochemistryMass SpectrometryAnalytical Chemistrychemistry.chemical_compoundCell Line TumorHumansIsoneorautenolCytotoxic T cellErythrinaErythrinaLupeolStigmasterolMolecular StructurebiologyPlant ExtractsOrganic ChemistryFabaceaeAntimicrobialbiology.organism_classificationAntineoplastic Agents PhytogenicAnti-Bacterial AgentschemistryCinnamatesPlant BarkDrug Screening Assays AntitumorDerivative (chemistry)Natural Product Research
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Effect of simulated gastrointestinal digestion on plant sterols and their oxides in enriched beverages

2013

Abstract This study evaluates the bioaccessibility (percentage of soluble compound available for absorption) of plant sterols (PS) and their oxides (phytosterol oxidation products, POPs) after simulated gastrointestinal digestion in fruit (Fb), milk (M) and fruit-based milk beverages with (FbM a ) or without (FbM b ) tangerine juice. In beverages and their bioaccessible fraction (BF), campesterol, campestanol, stigmasterol, β-sitosterol and sitostanol were detected. Bioaccessibility of total PS ranged between 2.62 and 6.48%, FbM b yielding the highest value, followed by FbM a  > Fb > M. Campesterol/campestanol were the most bioaccessible PS. Only oxides of β-sitosterol were detected in beve…

Absorption (pharmacology)StigmasterolChromatographyCampesterolPhytosterolBEVERAGESCampestanolPLANT STEROLchemistry.chemical_compoundchemistryPLANT STEROL; SIMULATED GASTROINTESTINAL DIGESTION; STEROL OXIDATION PRODUCTS; BEVERAGESFood scienceGas chromatography–mass spectrometrySolubilitySIMULATED GASTROINTESTINAL DIGESTIONPlant sterolsSTEROL OXIDATION PRODUCTSFood Science
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A new dibenzofuran and other constituents from Ligularia caloxantha, a Chinese medicinal plant.

2008

A new dibenzofuran named 1,2,4-trimethyl-7,8-dimethoxy-dibenzofuran (1), together with seven known compounds, euparin (2), 2,5-diacetyl-6-hydroxy-benzofuran (3), 2-acetyl-5,6-dimethoxy-benzofuran (4), gummosogenin (5), lupeol (6), stigmasterol (7) and (E)-2,5-dihydroxy-cinnamic acid (8), were isolated from the roots of Ligularia caloxantha, a Chinese medicinal plant. The structures of the compounds were elucidated by spectroscopic methods.

chemistry.chemical_classificationStigmasterolMolecular StructureChemistryOrganic ChemistryPlant ScienceLigularia caloxanthaAsteraceaeBiochemistryPlant RootsAnalytical ChemistryDibenzofuranchemistry.chemical_compoundTriterpeneOrganic chemistryBenzofuranLupeolBenzofuransDrugs Chinese HerbalNatural product research
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Wybrane fenomeny mistyczne w doświadczeniu religijnym Alicji Lenczewskiej w świetle jej pism

2019

Artykuł traktuje o polskiej nauczycielce, katoliczce, Alicji Lenczewskiej (1934-2012), poślubionej mistycznie Bogu, autorce dwutomowego dzieła, w którym utrwaliła pouczenia Zbawiciela, przedstawiła dzieje swojej duszy i opisała otrzymane od Stwórcy nadzwyczajne charyzmaty, do których należy zaliczyć: mistyczne zaślubiny, ekstazy, stygmaty niewidzialne i obrazy duchowe.

ekstazaobrazy duchoweZaślubiny mistycznestygmatyMystical marriagespiritual imagesecstasystigmasStudia Paradyskie
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Contribution à l’étude de la fraction insaponifiable de trois huiles d’olive issues des variétés Guasto, Rougette et Blanquette plantés dans l’est al…

2010

The sterol profile of three Algerian virgin olive oils produced from Guasto, Blanquette and Rougette cultivar’s, varieties grown in the East of the country, was established by gas chromatography using a flame ionization detector and coupled to mass spectrometry. Four sterol compounds were identified and characterized in the three oils which are, sitosterol always predominant (43-66%), delta 5-avenasterol (8-13%), stigmasterol (≤ 1,5%) and campesterol (1-2%); one methyl sterol (4-methylsterol) : citrostadienol (4-7%) and two triterpenic alcohols : 24-methylene cycloartanol (10-33%) and cycloartenol (3-13%). These results vary according to campany and variety. Our study shows that most of the…

StigmasterolChromatographyCampesterolphytosterolslcsh:TP670-699Mass spectrometryolive oilBiochemistrySterollaw.inventionchemistry.chemical_compoundchemistrylawCycloartenolcultivarsFlame ionization detectorCultivarGas chromatographylcsh:Oils fats and waxesOlea europaeaFood ScienceOléagineux, Corps gras, Lipides
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An expeditious synthesis of spinasterol and schottenol, two phytosterols present in argan oil and in cactus pear seed oil, and evaluation of their bi…

2015

International audience; Spinasterol and schottenol, two phytosterols present in argan oil and in cactus pear seed oil, were synthesized from commercially available stigmasterol by a four steps reactions. In addition, the effects of these phytosterols on cell growth and mitochondrial activity were evaluated on 158N murine oligodendrocytes, C6 rat glioma cells, and SK-N-BE human neuronal cells with the crystal violet test and the MTT test, respectively. The effects of spinasterol and schottenol were compared with 7-ketocholesterol (71CC) and ferulic acid, which is also present in argan and cactus pear seed oil. Whatever the cells considered, dose dependent cytotoxic effects of 71CC were obser…

Central Nervous Systemfood.ingredientCrystal violet testClinical BiochemistryStigmasterol[ PHYS.COND.CM-MS ] Physics [physics]/Condensed Matter [cond-mat]/Materials Science [cond-mat.mtrl-sci]Argan oilOrganic synthesisBiologyBiochemistryCell LineFerulic acidPyruschemistry.chemical_compoundMiceEndocrinologyfoodSchottenolCytotoxic T cellAnimalsHumansPlant OilsMolecular BiologySpinasterolCell ProliferationPharmacologyPEARMIT testStigmasterolCell growthOrganic ChemistryPhytosterolsNervous cellsSitosterolsMitochondriaRatsSpinasterolchemistryBiochemistryCactusSeeds
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