Search results for "SAP"

showing 10 items of 1142 documents

Steroidal saponins from Dioscorea preussii.

2014

Abstract Three new steroidal saponins, named diospreussinosides A–C (1–3), along with two known ones (4, 5) were isolated from rhizomes of Dioscorea preussii. Their structures were elucidated mainly by 1D and 2D NMR spectroscopic analysis and mass spectrometry as (25S)-17α,25-dihydroxyspirost-5-en-3β-yl-O-α- l -rhamnopyranosyl-(1 → 4)-α- l -rhamnopyranosyl-(1 → 4)-β- d -glucopyranoside (1), (25S)-17α,25-dihydroxyspirost-5-en-3β-yl-O-α- l -rhamnopyranosyl-(1 → 4)-α- l -rhamnopyranosyl-(1 → 4)-[α- l -rhamnopyranosyl-(1 → 2)]-β- d -glucopyranoside (2), and (24S,25R)-17α,24,25-trihydroxyspirost-5-en-3β-yl-O-α- l -rhamnopyranosyl-(1 → 4)-α- l -rhamnopyranosyl-(1 → 4)-[α- l -rhamnopyranosyl-(1 → …

PharmacologyDioscorea preussiiMolecular StructureStereochemistryChemistryDioscoreaPhytosterolsGeneral MedicineSaponinsMass spectrometryHCT116 CellsRhizomeDihydroxylationCarcinoma CellDrug DiscoveryHumansDrug Screening Assays AntitumorCytotoxicityTwo-dimensional nuclear magnetic resonance spectroscopyHT29 CellsHuman colonFitoterapia
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Eight-week consumption of milk enriched with omega 3 fatty acids raises their blood concentrations yet does not affect lipids and cardiovascular dise…

2014

Adequate concentrations of omega 3 fatty acids (FA) may be maintained by consuming foods naturally rich in or functional foods enriched with those essential FA. We assessed the effects of an 8-week consumption of milk enriched with 400. mg of omega 3 FA on blood lipid levels and selected cardiovascular risk factors in adult healthy volunteers. Participants (n= 157) were randomized to consume - for eight weeks - either 500. mL/day of 1% fat milk providing 150. mg of eicosapentaenoic (EPA), 150. mg of docosahexaenoic (DHA), and 100. mg of α-linolenic (ALA) acids or 500. mL/day of non-enriched 1% fat milk. At week 8, we observed significant increments of blood EPA and DHA in the intervention g…

PharmacologyEicosapentaenoic acidmedicine.diagnostic_testHomocysteineBlood lipidsPhysiologyMilk enriched with fish oilBiologyEicosapentaenoic acidLeukotriene B4Thromboxane B2Thromboxane B2chemistry.chemical_compoundDocosahexaenoic acidchemistryDocosahexaenoic acidHealthy volunteersmedicineDisease riskOmega 3 fatty acidPharmacology (medical)Food scienceLipid profileDocosahexaenoic acid; Eicosapentaenoic acid; Leukotriene B4; Milk enriched with fish oil; Omega 3 fatty acids; Thromboxane B2; Pharmacology; Pharmacology (medical); Food ScienceFood Science
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A review of the pharmacology and toxicology ofAstragalus

1997

Some Astragalus species are used as forage for livestock and wild animals. Many species are used in folk medicine for their hepatoprotective, antioxidative, immunostimulant, and antiviral properties, whereas others are toxic, and in many cases the toxic principles can pass to humans through milk and meat. Three groups of chemicals have been described as pharmacologically active principles: polysaccharides, saponins and phenolics. In addition, three kinds of toxic principles have been reported: indolizidine alkaloids, aliphatic nitro compounds and selenium. © 1997 John Wiley & Sons, Ltd.

PharmacologyFolk medicinechemistry.chemical_classificationAstragalus speciesAlkaloidSaponinfood and beveragesIndolizidineBiological activityBiologyPharmacognosybiology.organism_classificationToxicologychemistry.chemical_compoundAstragaluschemistryPhytotherapy Research
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Selektionstheorie und Rassenbildung beim Menschen

1952

So far, the applications of the theory of selection to human race formation have primarily considered the selective quality of individual race characters which are preferred by classification. However only few physiologically important race characters have been found to have an evident selective advantage. It is the climate laws, however, that prompt the assumption that selection will take place according to differences of vitality and fertility under certain climatic conditions and that the visible race characters are but incidental effects of pleiotropic gene. It also appears that, in contrast to selection, mutability must be given more consideration to-day than before. For instance the e…

PharmacologyGeneticsCell BiologyBiologyVitalityCellular and Molecular NeuroscienceTime factorRace (biology)Evolutionary biologyHomo sapiensSelective advantageMolecular MedicineQuality (philosophy)Molecular BiologySelection (genetic algorithm)Experientia
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Steroidal saponins from Dracaena marginata

2013

Three new steroidal saponins and ten known ones were isolated from the bark of Dracaena marginata, along with two known steroidal saponins from the roots. Their structures were elucidated on the basis of extensive 1D and 2D NMR experiments and mass spectrometry as (25R)-26-(beta-D-glucopyranosyloxy)3beta,22alpha-dihydroxyfurost-5-en-1beta-yl O-alpha-L-rhamnopyranosyl-(1 --> 2)-[alpha-L-rhamnopyranosyl-(1 --> 4)]-beta-D-glucopyranoside (1), (25R)-26-(beta-D-glucopyranosyloxy)-3beta,22alpha-dihydroxyfurost-5-en-1beta-yl O-alpha-L-rhamnopyranosyl-(1 --> 2)-4-O-sulfo-alpha-L-arabinopyranoside (2), and (25S)-3beta-hydroxyspirost-5-en-1beta-yl O-alpha-L-rhamnopyranosyl-(1 --> 2)-4-O-sulfo-alpha-L…

PharmacologyMagnetic Resonance SpectroscopyTraditional medicinebiologyChemistryDracaena marginataPlant ScienceGeneral MedicineNuclear magnetic resonance spectroscopySaponinsMass spectrometrybiology.organism_classificationMiceAsparagaceaeComplementary and alternative medicinevisual_artCell Line TumorDrug Discoveryvisual_art.visual_art_mediumAnimalsHumansBarkTwo-dimensional nuclear magnetic resonance spectroscopyDracaenaDracaena
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Spirostane-Type Saponins from Dracaena fragrans Yellow Coast

2015

Three steroidal glycosides were isolated from the bark of Dracaena fragrans (L.) Ker Gawl. « Yellow Coast », and a fourth from the roots and the leaves. Their structures were characterized on the basis of extensive 1D and 2D NMR experiments and mass spectrometry, and by comparison with NMR data of the literature. These saponins have the spirostane-type skeleton and are reported in this species for the first time.

PharmacologyTraditional medicineSteroidal glycosidesDracaena fragransPhytosterolsPlant ScienceGeneral MedicineSaponinsBiologybiology.organism_classificationComplementary and alternative medicinevisual_artDrug Discoveryvisual_art.visual_art_mediumBarkDracaena
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Triterpenoid Saponins From the Root Bark of Haplocoelum congolanum

2019

Two undescribed triterpenoid saponins together with 5 known ones were isolated from the root bark of Haplocoelum congolanum Hauman. Their structures were elucidated by spectroscopic methods including one-dimensional and two-dimensional nuclear magnetic resonance experiments in combination with mass spectrometry as 3- O-(4- O-[3-hydroxy-3-methylglutaryl])-α-l-arabinopyranosyl-(1→3)-α-l-rhamnopyranosyl-(1→2)-[β-d-glucopyranosyl-(1→4)]-α-l-arabinopyranosyloleanolic acid and 3- O-α-l-arabinofuranosyl-(1→3)-α-l-rhamnopyranosyl-(1→2)-[β-d-glucopyranosyl-(1→4)]-α-l-arabinopyranosyloleanolic acid.

PharmacologybiologyTraditional medicine010405 organic chemistryChemistryPlant ScienceGeneral MedicineSapindaceaebiology.organism_classification01 natural sciences0104 chemical sciences010404 medicinal & biomolecular chemistryHaplocoelumTriterpenoidComplementary and alternative medicinevisual_artDrug Discoveryvisual_art.visual_art_mediumBarkNatural Product Communications
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Cycloartane-type saponins from astragalus tmoleus var. tmoleus

2016

Five known cycloartane-type glycosides were isolated from the roots of A. tmoleus Boiss. var. tmoleus. The identification of these compounds was mainly achieved by 1D and 2D NMR spectroscopic techniques and FABMS. The results of our studies confirm that triterpene saponins with the cycloartane-type skeleton might be chemotaxonomically significant for the genus Astragalus.

Pharmacologychemistry.chemical_classificationMagnetic Resonance SpectroscopybiologyTraditional medicinePlant roots010405 organic chemistryGlycosidePlant ScienceGeneral MedicineFabaceaeAstragalus PlantSaponinsbiology.organism_classification01 natural sciencesPlant Roots0104 chemical sciences010404 medicinal & biomolecular chemistryAstragalusComplementary and alternative medicinechemistryTriterpeneGenusDrug DiscoveryAstragalus Plant
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Triterpene Saponins from the Roots of Achyranthes bidentata

2001

Three saponins, oleanolic acid-28- O -s-D-glucopyranoside (1), chikusetsusaponin V (2), and 3- O -s-D-glucopyranosyl-oleanolic acid-28- O -s-D-glucopyranoside (3) were isolated from the roots of Achyranthes bidentata Blume (Amaranthaceae). No activity was shown in the granulocyte phagocytosis test nor in the test of the potentiation of the cytotoxicity of cisplatin in human colon cancer cells. This is the first report of compounds 1, 2 and 3 isolated from Achyranthes species. Furthermore, the NMR data of 2 completed the partially published data.

Pharmacologychemistry.chemical_classificationTraditional medicineSaponinPharmaceutical ScienceBiological activityGeneral MedicineAmaranthaceaeBiologybiology.organism_classificationIn vitroComplementary and alternative medicinechemistryTriterpeneDrug DiscoveryMolecular MedicineAchyranthesCytotoxicityAchyranthes bidentataPharmaceutical Biology
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Antiproliferative oleanane saponins from Polyscias guilfoylei

2008

Three new oleanane saponins (1–3), together with four known ones (4–7), were isolated from the aerial parts of Polyscias guilfoylei. Their structures were elucidated by 1D and 2D NMR experiments, including 1D TOCSY, DQF-COSY, ROESY, HSQC, and HMBC spectroscopy, as well as ESIMS analysis. The antiproliferative activity of all compounds was evaluated using three murine and human cancer cell lines; J774.A1, HEK-293, and WEHI-164. All the compounds were inactive except for 3β- O-[β-D-glucopyranosyl-(1→2)-α-L-arabinopyranosyl]-echinocystic acid 28-[ O-β-D-glucopyranosyl-(1→6) O-β-D-glucopyranosyl] ester (3), which was active against all the cell lines.

Pharmacologychemistry.chemical_classificationbiologyStereochemistryGlycosidePlant ScienceGeneral Medicinebiology.organism_classificationPolyscias guilfoyleiSettore CHIM/08 - Chimica FarmaceuticaOleanane Saponins Antiproliferative effectsTerpenechemistry.chemical_compoundComplementary and alternative medicinechemistryDrug DiscoverySettore BIO/14 - FarmacologiaTwo-dimensional nuclear magnetic resonance spectroscopyOleanane
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