Search results for "phosphonates"

showing 10 items of 210 documents

Separation of aminoalkanephosphonic acid enantiomers by indirect UV detection capillary electrophoresis with application of cyclodextrins.

2003

Indirect UV detection capillary electrophoresis (CE) was used for the separation of aminoalkanephosphonic acid (AP) enantiomers by applying commercially available cyclodextrins as chiral discriminators. The results show that the separation of the enantiomers depends on pH of the background electrolyte, the molar ratio of cyclodextrin to aminophosphonic acid, and on the type of the applied chiral selector. Optimization of process conditions allowed enantiomeric baseline separation or partial separation of 12 out of 14 alpha-aminophosphonic acids studied. This type of CE might therefore be successfully used for routine determination of enantiomeric purity of aminophosphonic acids.

aminophosphonic acidsClinical Biochemistrycapillary electrophoresisOrganophosphonatesElectrolyteBiochemistryindirect UV detectionAnalytical ChemistryCapillary electrophoresisMolar ratiopolycyclic compoundsheterocyclic compoundsAmineschemistry.chemical_classificationCyclodextrinsChromatographyCyclodextrinorganic chemicalsElectrophoresis CapillaryStereoisomerismHydrogen-Ion ConcentrationProcess conditionschemistrycyclodextrinUv detectionEnantiomerenantiomer separationElectrophoresis
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BIODEGRADACJA ZWIĄZKÓW FOSFONOWYCH PRZEZ GRZYBY

2020

Phosphonates are the group of organophosphorus compounds, which are characterized by the presence of covalent bond(s) between carbon and phosphorus atom in their structure. Both; the natural and synthetic phosphonic compounds, are encountered in various ecosystems, however because of their wide range of applications, the latter ones are considerably more frequently discussed. Regarding the broad spectrum of biological activity, capability to chelate metal cations and environmental stability of direct carbon to phosphorus bond under physiological conditions, phosphonic compounds found a variety of applications e.g. as pesticides, drugs, anticorrosive agents, additives to surfactants and flam…

biotransformacjagrzybyzwiązki fosfonowebiodegradacjaphosphonatesbiotransformationfungibiodegradationWiadomości Chemiczne
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Medication-Related Osteonecrosis of Jaws (MRONJ) Prevention and Diagnosis: Italian Consensus Update 2020

2020

The Medication-Related Osteonecrosis of Jaws (MRONJ) diagnosis process and its prevention play a role of great and rising importance, not only on the Quality of Life (QoL) of patients, but also on the decision-making process by the majority of dentists and oral surgeons involved in MRONJ prevention (primary and secondary). The present paper reports the update of the conclusions from the Consensus Conference—held at the Symposium of the Italian Society of Oral Pathology and Medicine (SIPMO) (20 October 2018, Ancona, Italy)—after the newest recommendations (2020) on MRONJ were published by two scientific societies (Italian Societies of Maxillofacial Surgery and Oral Pathology and Medicine, SI…

bisphosphonateOral SurgeonHealth Toxicology and Mutagenesislcsh:MedicineMRONJantiangiogenic agents; antiresorptive drugs; bisphosphonates; cancer; denosumab; dentistry; MRONJ; oral surgery; osteoporosis; prevention models; bisphosphonate-associated osteonecrosis of the jaw; bone density conservation agents; diphosphonates; humans; Italy; quality of life0302 clinical medicineprevention modelCancerantiangiogenic agentsdentistryBone Density Conservation AgentsDiphosphonatesConference ReportBisphosphonatesAntiresorptive DrugsDenosumabItaly030220 oncology & carcinogenesisBisphosphonate-Associated Osteonecrosis of the JawDenosumabmedicine.drugoral surgerymedicine.medical_specialtyOral surgery03 medical and health sciencesOral surgeryAntiangiogenic agentsOral and maxillofacial pathologymedicinecancerHumansantiangiogenic agentantiresorptive drugsIntensive care medicinePrevention modelsbisphosphonatesantiresorptive drugAntiangiogenic agentsbusiness.industrylcsh:RPublic Health Environmental and Occupational Healthdenosumab030206 dentistrymedicine.diseaseosteoporosisAntiresorptive drugsDentistryOsteoporosisprevention modelsbusinessAntiangiogenic agents; Antiresorptive drugs; Bisphosphonates; Cancer; Denosumab; Dentistry; MRONJ; Oral surgery; Osteoporosis; Prevention models
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Carboranylphosphinic Acids: A New Class of Purely Inorganic Ligands

2015

Purely inorganic carboranyl phosphinates were prepared, and the influence of the cluster on the reactivity of the phosphinate group was studied. Electron-withdrawal by the carboranyl carbon atoms, combined with space-filling efficiency and enhanced aromaticity of the cluster cage, renders the phosphorus more difficult to oxidize. This enables carboranyl phosphinates to survive harsh oxidizing conditions, a property which is uncommon in organic phosphinates.

carboranes010405 organic chemistryHydrogen bondOrganic Chemistryphosphonateschemistry.chemical_elementAromaticityGeneral ChemistryPhosphinatehydrogen bonding010402 general chemistry01 natural sciencesCatalysis0104 chemical scienceschemistryOxidizing agentCluster (physics)Organic chemistryReactivity (chemistry)ta116CarbonphosphinateshydrophobicityChemistry - A European Journal
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Determination of optical purity of phosphonic acid analogues of aromatic amino acids by capillary electrophoresis with alpha-cyclodextrin.

2000

A simple and efficient method for the determination of enantiomeric purity of structurally diverse phosphonic and phosphinic acid analogues of phenylalanine and phenylglycine using capillary electrophoresis is presented. These preliminary studies indicated that the enantiomer separation is strongly dependent on the structure of the aminophosphonic acid.

chemistry.chemical_classificationCyclodextrinsalpha-CyclodextrinsChromatographyCyclodextrinOrganic ChemistryOrganophosphonatesElectrophoresis CapillaryPhenylalanineGeneral MedicineBiochemistryAnalytical ChemistryAmino acidchemistry.chemical_compoundCapillary electrophoresischemistryBenzene derivativesAromatic amino acidsphosphonic acidsEnantiomerenantiomer separationAmino AcidsEnantiomeric excessJournal of chromatography. A
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Synthesis of N-methyl alkylaminomethane-1,1-diphosphonic acids and evaluation of their complex-formation abilities towards copper(II)

2015

Abstract A series of N -methyl alkylaminomethane-1,1-diphosphonic acids ( 3a – g ) with a common tertiary nitrogen atom (CH 3 –N–R) bearing linear or branched alkyl, cycloheptyl or phenylalkyl R substituents was synthesized in the reaction of diethylphosphonate with triethyl orthoformate and secondary amine followed by hydrolysis, and by the Eschweiler–Clarke methylation of the alkylaminomethane-1,1-diphosphonic acids with formic acid and formaldehyde. Complex-formation abilities of 3a – g towards copper(II) in solution were studied by means of pH-potentiometry, ESI-MS spectrometry, UV–Vis and EPR methods. Evaluation of stability constants for the Cu(II) complexes of 3a – g has revealed the…

chemistry.chemical_classificationSteric effectsVis spectroscopyFormic acidStereochemistryProtonationpH potentiometryTriethyl orthoformateMedicinal chemistrylaw.inventionInorganic Chemistrychemistry.chemical_compoundchemistrylawMaterials ChemistryElectronic effectCopper(II) complexesAmine gas treatingEPRPhysical and Theoretical ChemistryElectron paramagnetic resonancebisphosphonatesAlkylPolyhedron
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Herbicidally Active Derivatives of Aminomethylenebis-Phosphonic Acid-Mode of Action and Structure - Activity Relationship

1996

Abstract: (N-pyridylamino)methylenebisphosphonates exhibit strong herbicidal activity which may be reversed by supplementation of the growth media with aromatic amino acids. They appeare to be the inhibitors of aromatic amino acids biosynthesis acting as inhibitors of DAHP synthase the first enzyme of shikimate pathway. Over 40 analogues of these acids were synthesized in order to determine the structure-activity relationship.

chemistry.chemical_classificationamino acid biosynthesisbiologyStereochemistryOrganic Chemistry(N-pyridylamino)methylenebisphosphonatesDAHP synthaseBiochemistryInorganic Chemistrychemistry.chemical_compound(N-pyridylamino)methylenebisphosphonates; amino acid biosynthesis; inhibitorsEnzymechemistryBiosynthesisinhibitorsbiology.proteinAromatic amino acidsStructure–activity relationshipShikimate pathwayMode of actionPhosphorus, Sulfur, and Silicon and the Related Elements
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Separation of aromatic aminophosphonic acid enantiomers by capillary electrophoresis with the application of cyclodextrins

2002

The detailed studies concerning capillary electrophoresis separation of aminophosphonic acid enantiomers with various commercially available cyclodextrins are presented. The obtained results show that the separation of these stereoisomers is dependent on pH of background electrolyte, concentration of cyclodextrin as well as on the type of applied chiral selector. The separation mechanism is based on the co-operative effect of hydrogen bond type interactions enhanced by hydrophobic forces and sterical constrains between aminophosphonate and cyclodextrin. With application of elaborated method, enantiomeric baseline or partial separation of 18 alpha-aminophosphonic acids was achieved. This sep…

chemistry.chemical_classificationcyclodextrinsChromatographyaminophosphonic acidsCyclodextrinHydrogen bondOrganic ChemistryOrganophosphonatesElectrophoresis CapillaryStereoisomerismorganophosphorus compoundsGeneral MedicineElectrolyteBiochemistryAnalytical ChemistryHydrophobic effectCapillary electrophoresischemistryAminophosphonatePhase compositionpolycyclic compoundsEnantiomerJournal of Chromatography A
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Herbicidal Derivatives of Aminomethylenebisphosphonic Acid. Part IV. Hydroxyalkylidenebisphosphonates, Iminomethylenebisphosphonates and Ureidomethyl…

2000

Derivatives of aminomethylenebisphosphonic acids constitute a class of promising herbicides. Replacement of the amino group by hydroxyl, ureido, thioureido, or imino moieties leads to compounds of significant herbicidal properties. This indicates that protonated amino function is not a requirement for phytotoxic action of bisphosphonates.

chemistry.chemical_compoundglyphosateamino acid biosynthesisThioureaChemistryStereochemistryProtonationPlant SciencebisphosphonatesAgronomy and Crop ScienceJournal of Plant Growth Regulation
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Organophosphonate utilization by the wild‐type strain of cladosporium resinae

1997

We studied the biodegradation of compounds containing phosphorus‐to‐carbon bond by using wild‐type strain of Cladosporium resinae. The substrate specificity of the strain was studied and we found that it is able to utilize a range of structurally diverse organophosphonates as a sole source of phosphorus. This ability is inducible as indicated by the presence of a lag phase of the growth. A popular herbicide glyphosate is also degraded by the fungi. This indicates that Cladosporium resinae may play an important role in biodegradation of this herbicide. The strain which we used, however, did not metabolise any phosphonates when they served as the sole carbon or nitrogen sources.

ciliatineStrain (chemistry)biologyHealth Toxicology and MutagenesisPhosphoruschemistry.chemical_elementBiodegradationcarbon‐to‐phosphorus bondbiology.organism_classificationPollutionbiodegradationchemistry.chemical_compoundBiochemistrychemistryglyphosateGlyphosateHerbicide glyphosateEnvironmental ChemistryOrganophosphonatesCladosporiumWild type strainToxicological and Environmental Chemistry
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