Search results for "CoV"

showing 10 items of 9749 documents

A new electrophilic addition to acetylenes. Synthesis of 1,2-iodofunctionalized olefins

1986

Abstract Acetylenes react with bis(pyridine)iodo(I) tetrafluoroborate ( 1 ) in the presence of a wide variety of nucleophiles (F, Cl, Br, I, SCN, pyridine, OAc, anisole, H) to give 1,2-iodofunctionalized olefins ( 4 ).

Addition reactionTetrafluoroborateElectrophilic additionOrganic ChemistryHalocarbonAnisoleBiochemistryMedicinal chemistrychemistry.chemical_compoundchemistryNucleophileDrug DiscoveryPyridineOrganic chemistryAliphatic compoundTetrahedron Letters
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A new and versatile method for iodofunctionalization of 1,3-dienes

1986

Abstract We wish to report the reactions of conjugated dienes with I(py) 2 BF 4 . This simple and general method allows the regiospecific 1,2-addition of iodine and a nucleophile to terminal dienes and the 1,4-addition to internal dienes.

Addition reactionchemistry.chemical_compoundGeneral methodNucleophileChemistryOrganic ChemistryDrug DiscoveryPyridineHalogenationOrganic chemistryConjugated systemAliphatic compoundBiochemistryTetrahedron Letters
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1,4-regioselective iodofunctionalizations of 1,3-butadiene

1988

Abstract Addition reactions of benzene and acetonitrile to 1,3-butadiene are described. This new iodofunctionalization process proceeds “via” iodonium ion-allylic cation equilibrium and gives regioselectively 1,4-adducts, which can be alternatively obtained by acid treatment of the 1,2-derivative 8 .

Addition reactionchemistry.chemical_compoundchemistryOrganic ChemistryDrug DiscoveryRegioselectivityOrganic chemistry13-ButadieneAcid treatmentBenzeneAcetonitrileBiochemistryTetrahedron Letters
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Fine-needle biopsy of parathyroid adenomas

1986

High-resolution real-time sonography was performed in 15 cases of clinically and chemically suspected primary hyperparathyroidism and in 20 patients with different thyroid nodules. The suspected enlarged parathyroid glands and the thyroid nodules were percutaneously punctured under sonographic control. Concentrations of parathyroid hormone, human thyroglobulin, and human calcitonin were measured in the aspirate, and immunocytology was performed. The mean concentration of the aspirated parathyroid hormone in the parathyroid glands was 4,013.6 pmol/l +/- 4,519 (SD) as compared with 14.9 pmol/l +/- 8.7 in the thyroid nodules. Thyroglobulin was present in the aspirated fluid of parathyroid aden…

AdenomaAdultMaleThyroid nodulesendocrine systemPathologymedicine.medical_specialtyendocrine system diseasesAdenomamedicine.medical_treatmentFluorescent Antibody TechniqueParathyroid hormoneParathyroid GlandsDrug DiscoverymedicineHumansGenetics (clinical)AgedUltrasonographyHyperparathyroidismParathyroid neoplasmbusiness.industryBiopsy NeedleThyroidGeneral MedicineMiddle Agedmedicine.diseaseParathyroid Neoplasmsmedicine.anatomical_structureParathyroid HormoneMolecular MedicineFemaleThyroglobulinbusinesshormones hormone substitutes and hormone antagonistsPrimary hyperparathyroidismKlinische Wochenschrift
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Hypermineralocorticoidism and hypertension

1971

Die mit Hypokaliamie, Uberproduktion von Mineralocorticoiden (Aldosteron und/oder Corticosteron und Desoxycorticosteron) und Aktivitatsanderungen des Renin-Angiotensinsystems einhergehenden Hochdrucksformen werden beschrieben. Sie lassen sich nach willkurlich gewahlten biochemischen Kriterien in drei Gruppen einteilen: a) Hypermineralocorticoidismus mit Reninsuppression und Aldosteronismus, b) Hypermineralocorticoidismus mit Reninund Aldosteronsuppression und c) Hypermineralocorticoidismus mit erhohtem Plasmarenin und Aldosteronismus. Jede dieser Gruppen besteht aus mehreren Syndromen, die sich durch ihr adrenocorticales Sekretionsmuster und/oder ihre morphologischen Nebennierenrindenverand…

AdenomaGynecologymedicine.medical_specialtyAdrenocortical HyperfunctionHyperplasiabusiness.industryAdrenal Gland NeoplasmsHypokalemiaGeneral MedicineRenal Artery ObstructionDexamethasoneDiagnosis DifferentialHypertension MalignantMineralocorticoidsHyperaldosteronismHypertensionReninDrug DiscoverymedicineHumansMolecular MedicinebusinessAldosteroneCushing SyndromeGenetics (clinical)Klinische Wochenschrift
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Fluorescent Probes for Ecto-5′-nucleotidase (CD73)

2020

[Image: see text] Ecto-5′-nucleotidase (CD73) catalyzes the hydrolysis of AMP to anti-inflammatory, immunosuppressive adenosine. It is expressed on vascular endothelial, epithelial, and also numerous cancer cells where it strongly contributes to an immunosuppressive microenvironment. In the present study we designed and synthesized fluorescent-labeled CD73 inhibitors with low nanomolar affinity and high selectivity based on N(6)-benzyl-α,β-methylene-ADP (PSB-12379) as a lead structure. Fluorescein was attached to the benzyl residue via different linkers resulting in PSB-19416 (14b, K(i) 12.6 nM) and PSB-18332 (14a, K(i) 2.98 nM) as fluorescent high-affinity probes for CD73. These compounds …

Adenosinemedicine.medical_treatmentInflammation01 natural sciencesBiochemistryecto-5′-nucleotidaseHydrolysisDrug Discoverymedicine010405 organic chemistryChemistryfungiOrganic ChemistryEcto 5 nucleotidase cd73ImmunotherapyAdenosineFluorescence0104 chemical sciences010404 medicinal & biomolecular chemistryBiochemistryCancer cellCD73fluorescenceimmunotherapymedicine.symptominflammation.medicine.drugACS Medicinal Chemistry Letters
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Current dental adhesives systems. A narrative review.

2012

Adhesive dentistry is based on the development of materials which establish an effective bond with the tooth tissues. In this context, adhesive systems have attracted considerable research interest in recent years. Successful adhesive bonding depends on the chemistry of the adhesive, on appropriate clinical handling of the material as well as on the knowledge of the morphological changes caused on dental tissue by different bonding procedures. This paper outlines the status of contemporary adhesive systems, with particular emphasis on chemical characteristics and mode of interaction of the adhesives with enamel and dentinal tissues. Dental adhesives are used for several clinical application…

Adhesive bondingPolyurethanesAcrylic ResinsDentistryDental CementsComposite ResinsComposite resinstomatognathic systemSettore MED/28 - Malattie OdontostomatologicheDrug DiscoveryAdhesive systemHumansDental EtchingDental EnamelPharmacologyOrthodonticsEnamel paintbusiness.industryDentineDental BondingDental Adhesivesstomatognathic diseasesEnamelvisual_artDentin-Bonding AgentsDental EtchingDentinvisual_art.visual_art_mediumNarrative reviewAdhesivebusinessDental adhesivePhosphoric acidCurrent pharmaceutical design
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Effect of the basidiomycete Poria cocos on experimental dermatitis and other inflammatory conditions.

1997

The hydroalcoholic extract from P. cocos was examined for oral and topical anti-inflammatory activities. It proved to be active against carrageenan, arachidonic acid, tetradecanoyl phorbol acetate (TPA) acute edemas, TPA chronic inflammation and oxazolone delayed hypersensitivity in mice. Two lanostane-type triterpenes were isolated and identified by spectroscopic methods as dehydrotumulosic and pachymic acids. Their ID50 on acute TPA edema was 4.7 x 10(-3) and 6.8 x 10(-4) mumol/ear, respectively.

Administration TopicalAnti-Inflammatory AgentsAdministration OralDermatitisPharmacognosyPharmacologyCarrageenanOxazolonechemistry.chemical_compoundMiceEdemaDrug DiscoverymedicineAnimalsInflammationArachidonic Acidintegumentary systemPlant ExtractsBasidiomycotaGeneral ChemistryGeneral MedicineTriterpenesCarrageenanchemistryDelayed hypersensitivityTetradecanoylphorbol AcetateImmunologyPhorbolTetradecanoylphorbol AcetateArachidonic acidFemalemedicine.symptomChemicalpharmaceutical bulletin
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Topical anti-inflammatory activity of some Asian medicinal plants used in dermatological disorders.

2001

The topical anti-inflammatory activity of extracts from Cassia angustifolia, Rheum palmatum, Coptis chinensis, Phellodendron amurense and Scutellaria baicalensis, plants used in traditional East Asian medicine against different skin disorders, was studied. Though in different degree, all the extracts significantly inhibited the edema induced by 12-O-tetradecanoylphorbol-13-acetate (TPA), in both single or multiple application, oxazolone, and arachidonic acid (AA). None of the extracts inhibited in vitro the activity of phospholipase A(2) (PLA(2)) from Naja naja.

Administration TopicalAnti-Inflammatory AgentsPharmacognosyCassia angustifoliaPhospholipases Alaw.inventionMicelawCassiaDrug DiscoveryMedicineAnimalsEdemaRosalesPharmacologyRheum palmatumPlants MedicinalTraditional medicinebiologybusiness.industryOxazoloneGeneral MedicineCoptis chinensisbiology.organism_classificationPolygonaceaePhellodendron amurenseScutellaria baicalensisFemalebusinessPhytotherapyDrugs Chinese HerbalFitoterapia
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Viral exanthema as manifestation of SARS-CoV-2 infection

2020

Abstract Rationale: The clinical manifestations of the SARS-CoV-2 infection are mainly respiratory but the virus can cause a variety of symptoms. Dermatological findings are less well-characterized. Data is scarce on their timing, type and correlation with the immune response. Patient concerns: We present the case of SARS-CoV-2 infection in a previously healthy woman who presented with respiratory symptoms and developed anosmia, diarrhea, and an erythematous maculo-papular rash on day 15 from symptom onset. Diagnosis: The nasopharyngeal swab tested by real time PCR for COVID-19 was positive. We interpreted this as a viral exanthema likely caused by an immune response to SARS-CoV-2 nucleotid…

Administration TopicalvirusesAzithromycinAzithromycinLopinavirimmune responseCOVID-19 Testing0302 clinical medicine030212 general & internal medicineclinical manifestations4900virus diseasesLopinavirGeneral MedicineRashDrug CombinationsDiarrheaTreatment Outcome030220 oncology & carcinogenesisFemaleSymptom Assessmentmedicine.symptomCoronavirus InfectionsHydroxychloroquineResearch Articlemedicine.drugAdultmedicine.medical_specialtyPneumonia ViralAnosmiaAntiviral AgentsBetacoronavirus03 medical and health sciencesImmune systemImmunitymedicineHumansClinical Case ReportGlucocorticoidsPandemicsRitonavirClinical Laboratory TechniquesSARS-CoV-2business.industryfungiCOVID-19HydroxychloroquineExanthemabiochemical phenomena metabolism and nutritionDermatologybusinessanosmiaMedicine
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